Synthesis of optically pure 2-Aziridinemethanols: Versatile synthetic building blocks

DOI: 10.1248/cpb.42.2241

Source and publish data:

Chemical and Pharmaceutical Bulletin p. 2241 - 2250 (1994)

Update date:2022-09-26

Topics:

Authors:

Fujii Fujii

Nakai Nakai

Habashita

Hotta Hotta

Tamamura

Otaka Otaka

Ibuka Ibuka

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Article abstract of DOI:10.1248/cpb.42.2241

Synthesis of three cis-trans pairs of N-sulfonylated-2-aziridinemethanols starting from (S)-threonine, (R)-allothreonine, a chiral 2-amino alcohol, or enantiomerically enriched 2,3-epoxy alcohols is described. A synthetic route to N-tosyl- and N-mesyl-2-a

Full text of DOI:10.1248/cpb.42.2241

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