1-(phenylsulfonyl)indol-2-yl triflate: A versatile reagent for the synthesis of 2-substituted indoles

Article abstract of DOI:10.1080/00397919608004639

The palladium-catalysed reaction of 1-(phenylsulfonyl)indol-2-yl triflate 1 with a variety of aryl and heteroaryl boronic acids 2 or vinyl tributylstannane 3 provides a general and an efficient method for the synthesis of 2-substituted indoles 4.

Full text of DOI:10.1080/00397919608004639

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Synthetic Communications: An
International Journal for Rapid
Communication of Synthetic
Organic Chemistry
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1-(Phenylsulfonyl)indol-2-yl
Triflate: A Versatile Reagent for
the Synthesis of 2-Substituted
Indoles
Beno[icaron]t Joseph a , Béatrice Malpel a & Jean-
Yves Mérour a
a Institut de Chimie Organique et Analytique,
Université d'Orléans , BP 6759, 45067 ORLEANS
Cédex 2, France
Published online: 21 Aug 2006.
To cite this article: Beno[icaron]t Joseph , Béatrice Malpel & Jean-Yves Mérour
(1996) 1-(Phenylsulfonyl)indol-2-yl Triflate: A Versatile Reagent for the Synthesis
of 2-Substituted Indoles, Synthetic Communications: An International Journal for
Rapid Communication of Synthetic Organic Chemistry, 26:17, 3289-3295, DOI:
10.1080/00397919608004639
To link to this article: http://dx.doi.org/10.1080/00397919608004639
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