Efficient two-step synthesis of sulfonylguanidines from sulfonamides

Article abstract of DOI:10.1080/00397919608003832

Various sulfonylguanidines have been synthesized from a sulfonamide by two mild and efficient synthetic methods. In route A, the methylthio group of S-methylsulfonylisothiourea is displaced by a variety of amines while in route B the amines are reacted wi

Full text of DOI:10.1080/00397919608003832

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Synthetic Communications: An
International Journal for Rapid
Communication of Synthetic
Organic Chemistry
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Efficient Two-Step Syntheses
of Sulfonylguanidines from
Sulfonamides
Pierre Deprez a & Jean-Paul Vevert a
a Hoechst Marion Roussel, Centre de Recherches
Roussel Uclaf, 102 route de Noisy, 93235, Romaiville,
Cedex
Published online: 23 Aug 2006.
To cite this article: Pierre Deprez & Jean-Paul Vevert (1996) Efficient Two-Step
Syntheses of Sulfonylguanidines from Sulfonamides, Synthetic Communications: An
International Journal for Rapid Communication of Synthetic Organic Chemistry, 26:23,
4299-4310
To link to this article: http://dx.doi.org/10.1080/00397919608003832
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