A highly stereoselective synthesis of the functionalized (E)-alkene dipeptide isostere of Trp-Val via organocyanocopper-Lewis acid mediated reaction

DOI: 10.1248/cpb.45.1259

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Chemical and Pharmaceutical Bulletin p. 1259 - 1264 (1997)

Update date:2022-07-30

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Authors:

Noda, Masaki

Ibuka, Toshiro

Habashita, Hiromu

Fujii, Nobutaka

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Article abstract of DOI:10.1248/cpb.45.1259

A stereocontrolled synthesis of the (e)-alkene dipeptide isostere of Trp-Val is described. The stereospecific α-alkylation of the δ-amino-γ- mesyloxy-α,β-unsaturated ester via the organocyanocopper-Lewis acid mediated reaction, based on 1,3-transfer of ch

Full text of DOI:10.1248/cpb.45.1259

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