Serine derived NK1 antagonists 2: A pharmacophore model for arylsulfonamide binding

DOI: 10.1016/S0960-894X(98)00319-9

Source and publish data:

Bioorganic and Medicinal Chemistry Letters p. 1851 - 1856 (1998)

Update date:2022-08-05

Topics:

Authors:

Elliott Elliott

Broughton

Cascieri

Chicchi Chicchi

Huscroft

Kurtz Kurtz

MacLeod MacLeod

Sadowski

Stevenson

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Article abstract of DOI:10.1016/S0960-894X(98)00319-9

Modifications to the spirocyclic aryl sulfonamide portion of serine derived NK₁ antagonists allow a partial pharmacophore model to be developed.

Full text of DOI:10.1016/S0960-894X(98)00319-9

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