Preparation of fluorinated phenoxathiin dioxide monoamine oxidase-A inhibitors: Intramolecular radical substitution at sulfur versus the Mauthner synthesis

DOI: 10.1002/jhet.5570350332

Source and publish data:

Journal of Heterocyclic Chemistry p. 699 - 706 (1998)

Update date:2022-07-29

Topics:

Authors:

Boros, Eric E.

Hall, William R.

Harfenist, Morton

Kelley, James L.

Reeves, Mark D.

Styles, Virgil L.

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1002/jhet.5570350332

Five unique fluorinated analogs, 8a-c and 15a,b, of the monoamine oxidase-A inhibitor 3-iso-propoxyphenoxathiin 10,10-dioxide (II) were prepared via oxidation of the corresponding phenoxathiins 7 and 14. 3- Fluoro-7-isopropoxy- 7a, 2-fluoro-3-isopropoxy-

Full text of DOI:10.1002/jhet.5570350332

Products guided by the article

Product name:Phenol, 2-mercapto-5-(1-methylethoxy)-

Cas No:205187-15-1

R&D Labs maybe for 205187-15-1

Jiaxing Carry Bio-Chem Technology Co.,Ltd

website:http://www.carrybiotech.com

Contact:0573-82788958

Address:Add.Fl 3th, Pharm Vally,Kaichuang Rd, Xiuzhou District, Jiaxing, Zhejiang,314031,China
NIGNXIA XINDACHANG TECHNOLOGY CO.,LTD

Contact:86-0951-7815345

Address:North side of Qiyuan Road, west side of Yuanfeng Highway, New Material Park, Ningdong Energy and Chemical Industry Base, Ningxia,China
Tianjin Bright Future Technology Co., Ltd

Contact:0086-22-58016666

Address:NO.136 DongTeng Lake Street Tianjin Economic and Technology Development Area,Tainjin,China
Yingkou Sanzheng New Technology Chemical Industry Co., Ltd.

Contact:+86-417-2927806

Address:yingkou
Shijiazhuang Haotian Chemical Co., Ltd.

Contact:86-311-85044374

Address:293 Donggang Road

Relevant to this article

Concise and versatile syntheses of N-arylalkylpiperidines as potential intermediates for 4-anilidopiperidine analgesics

Doi:10.3987/COM-97-8056
(1998)
Reversible and irreversible inhibitory activity of succinic and maleic acid derivatives on acetylcholinesterase

Doi:10.1016/S0928-0987(03)00023-X
(2003)
Perfluoroalkyl- and perfluoroalkylether-substituted aromatic phosphates and phosphonates

Doi:10.1016/S0022-1139(98)00114-6
(1998)
The First Catalytic Asymmetric Allylation of Imines with the Tetraallylsilane-TBAF-MeOH System, Using the Chiral Bis-π-allylpalladium Complex

Doi:10.1021/jo035453b
(2004)
C-3- and C-4-alkylated polyhydroxypyrrolidines: Enantiospecific syntheses and glycosidase inhibitory activity

Doi:10.1021/jo980078m
(1998)
An enantioselective synthesis of (+)-pseudohygroline

Doi:10.1016/S0040-4039(98)00253-6
(1998)

Article Doi