
Bioorganic and Medicinal Chemistry Letters p. 3127 - 3132 (1998)
Update date:2022-07-30
Topics:
Darrow, James W.
Hadac, Elizabeth M.
Miller, Laurence J.
Sugg, Elizabeth E.
Incorporation of photolabile benzoyl (2a-d) or trifluoromethyl-3H- diazirine (3a-d) substituents into 1,5-benzodiazepine ligands did not significantly impair the rat CCK-A binding affinity of either agonists or antagonists. The modified agonist ligands al
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