European Journal of Medicinal Chemistry p. 447 - 455 (2013)
Update date:2022-08-03
Topics:
Shao, Hao
Shi, Shenhua
Foley, David W.
Lam, Frankie
Abbas, Abdullah Y.
Liu, Xiangrui
Huang, Shiliang
Jiang, Xiangrui
Baharin, Nadiah
Fischer, Peter M.
Wang, Shudong
A series of 2,4,5-trisubstituted pyrimidines have been synthesised and characterised, which exhibited potent CDK inhibition and anti-proliferative activities. The structure-activity relationship is analysed and a rational for CDK9 selectivity is discussed
View MoreTAIZHOU XINGCHENG CHEMPHARM CO.,LTD.
Contact:0086-0576-88551200,88886292 ,88880039
Address:B Area. 10 Floor.Yaodadasha. 289#.Shifu Road.Taizhou.Zhejiang.China
Jinan Jiaquan Chemical Co.,Ltd
Contact:+86-531-62318366
Address:Room 502 of Yidonghuayuan No.601 Huaxin Road Licheng District Jinan China
Shanghai shibo Chemical Co., Ltd
Contact:+86-021-60753516
Address:688 Qiushi Road, Jinshan High-tech Park, Shanghai, China,201512
Suzhou Ryan Pharmachem Technology Co.,Ltd
Contact:+86-0512-68780025
Address:B-301,No.2 Taishan Road,Suzhou New District,Jiangsu,P.R. China
Shanghai Yolne Chemical Co., Ltd
Contact:+86-21-62960152,61525205,61538832,61538837
Address:Floor 4,building 2, No. 3377, Kangxi Road, Pudong New District, Shanghai, China
Doi:10.1021/op2001723
(2011)Doi:10.1016/j.tet.2013.05.102
(2013)Doi:10.1021/acs.joc.5b01850
(2015)Doi:10.1016/S0020-1693(00)82342-7
(1984)Doi:10.1007/BF00807163
(1995)Doi:10.1134/S1070428006060248
(2006)