Rearrangement of primary 2,3-epoxy amines into 1,2-aziridinyl 3-ols

DOI: 10.1016/S0040-4039(00)79090-3

Source and publish data:

Tetrahedron Letters p. 5351 - 5354 (1992)

Update date:2022-08-04

Topics:

Authors:

Najime Najime

Pilard Pilard

Vaultier

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Article abstract of DOI:10.1016/S0040-4039(00)79090-3

Conditions were found to transform primary 2,3-epoxy amines into 1,2-aziridinyl 3-ols which involve an intramolecular opening of the epoxide ring mediated by trimethylaluminum.

Full text of DOI:10.1016/S0040-4039(00)79090-3

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