MONITORED AMINOLYSIS OF 3-ACYL-1,3-THIAZOLIDINE-2-THIONE WITH AMINO ACID AND ITS DERIVATIVE: PEPTIDE BOND FORMATION, CHEMOSELECTIVE ACYLATION, AND BRIDGING REACTION

DOI: 10.1246/cl.1981.463

Source and publish data:

Chemistry Letters p. 463 - 466 (1981)

Update date:2022-08-05

Topics:

Authors:

Nagao, Yoshimitsu

Miyasaka, Tadayo

Seno, Kaoru

Yagi, Masahiro

Fujita, Eiichi

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Article abstract of DOI:10.1246/cl.1981.463

As a new extention of the monitored aminolysis of 3-acyl-1,3-thiazolidine-2-thione, its applications to peptide bond formation, chemoselective acylation of amino acid, and bridging reaction on the enzyme model are reported.

Full text of DOI:10.1246/cl.1981.463

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