Bioorganic and Medicinal Chemistry Letters p. 4284 - 4287 (2011)
Update date:2022-07-29
Topics:
Watson, Christine
Owen, Dafydd R.
Harding, Denise
Kon-I, Kana
Lewis, Mark L.
Mason, Helen J.
Matsumizu, Miyako
Mukaiyama, Takasuke
Rodriguez-Lens, Margarita
Shima, Akiko
Takeuchi, Mifune
Tran, Isabelle
Young, Tim
A series of benzimidazole CB2 receptor agonists were prepared and their properties investigated. Optimisation of the three benzimidazole substituents led to the identification of compound 23, a potent CB2 full agonist (EC50 View More
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