Journal of Medicinal Chemistry p. 7555 - 7568 (2017)
Update date:2022-08-29
Topics:
Xia, Lizi
Burger, Wessel A. C.
Van Veldhoven, Jacobus P. D.
Kuiper, Boaz J.
Van Duijl, Tirsa T.
Lenselink, Eelke B.
Paasman, Ellen
Heitman, Laura H.
Ijzerman, Adriaan P.
We expanded on a series of pyrido[2,1-f]purine-2,4-dione derivatives as human adenosine A3 receptor (hA3R) antagonists to determine their kinetic profiles and affinities. Many compounds showed high affinities and a diverse range of k
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