
Journal of Heterocyclic Chemistry p. 839 - 843 (1990)
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The syntheses of 6-fluoro-7-piperazin-l-yl-9-cyclopropyl (or 9-p-fluorophenyl)-2,3,4,9- tetrahydroisothiazolo[5,4-b]quinoline-3,4-diones as well as novel synthesis of isothiazolo-3(2H)-one system are described. Key steps include the regiospecific displace
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()Doi:10.1021/jo00237a035
(1988)