Bioorganic and Medicinal Chemistry Letters p. 2340 - 2343 (2010)
Update date:2022-08-04
Topics:
Rimland, Joseph
Dunne, Angela
Hunjan, Suchete S.
Sasse, Rosemary
Uings, Iain
Montanari, Dino
Caivano, Matilde
Shah, Poonam
Standing, David
Gray, David
Brown, David
Cairns, William
Trump, Ryan
Smith, Paul W.
Bertheleme, Nicolas
D'Alessandro, Pier
Gul, Sheraz
Vimal, Mythily
Smith, David N.
Watson, Stephen P.
The identification of novel, potent, non-steroidal/small molecule functional GR antagonist GSK1564023A selective over PR is described. Associated structure-activity relationships and the process of optimisation of an initial HTS hit are also described.
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