
Journal of Medicinal Chemistry p. 1855 - 1859 (1991)
Update date:2022-08-03
Topics:
Glennon, Richard A.
Ismaiel, Abd M.
Smith, J. Doyle
Yousif, Mamoun
El-Ashmawy, Mahmoud
et al.
Certain benzomorphans, such as N-allylnormetazocine, are classical "?-opiates" that bind both at ? and phencyclidine (PCP) binding sites with modest affinity.Recently, we identified N-substituted 2-phenylaminoethane as being the primary ?-pharmacophore of
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