Studies in macrolide synthesis: A stereocontrolled synthesis of a (9S)-macrolide intermediate for oleandomycin using chiral boron reagents

DOI: 10.1016/S0040-4039(00)91728-3

Source and publish data:

Tetrahedron Letters p. 1767 - 1770 (1992)

Update date:2022-08-03

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Authors:

Paterson

Lister Lister

Norcross

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Article abstract of DOI:10.1016/S0040-4039(00)91728-3

The (9S)-macrolide 1 (P = TBS) was prepared in 14 stpes (5% yield) with 63% overall ds starting from the ethyl ketone (S)-2. The C₁-C₇ and C₈-C₁₃ segments, 3 and 4, were obtained via boron enolate aldol reaction

Full text of DOI:10.1016/S0040-4039(00)91728-3

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