Journal of labelled compounds and radiopharmaceuticals p. 363 - 368 (1997)
Update date:2022-08-03
Topics:
Matsuoka, Hiroharu
Kuroki, Toshio
Yano, Keiichi
Takeda, Yasuhisa
Synthesis of tritiated N-[4-(2,4-diaminopteridine-6-methyl)-3,4-dihydro-2H-1,4-benzothiazine-7 -carbonyl]-L-homoglutamic acid, [9-3H,]MX-68 (3), is described. [9-3H1MX-68 (3) was prepared via tritiation at the carbonyl group in 2,4-bis(butanoylamino)-6-formylpteridine (7) with sodium borotritiide.
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