
Chemical and Pharmaceutical Bulletin p. 1293 - 1299 (1997)
Update date:2022-08-04
Topics:
Okada, Minoru
Yoden, Toru
Kawaminami, Eiji
Shimada, Yoshiaki
Kudoh, Masafumi
Isomura, Yasuo
In order to study the potency of the 5-aminopyrimidine skeleton as an aromatase inhibitor, we synthesized various N,N-disubstituted-15- aminopyrimidine derivatives and evaluated their aromatase-inhibitory activity (in vitro) and their inhibitory activity
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