Highly stereocontrolled synthesis of enantiomeric 4-methoxy trinems via resolution of scalemic enol phosphates

DOI: 10.1016/0957-4166(96)00384-9

Source and publish data:

Tetrahedron Asymmetry p. 2929 - 2938 (1996)

Update date:2022-08-04

Topics:

Authors:

Panunzio, Mauro

Camerini, Roberto

Pachera, Roberta

Donati, Daniele

Marchioro, Carla

Perboni, Alcide

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Article abstract of DOI:10.1016/0957-4166(96)00384-9

Stereocontrolled syntheses of 4-methoxy trinem 2 and its enantiomer 3 were achieved using the ester enolate N-trimethylsilylimine approach. The key step was the resolution of racemic enolphosphates derived from ephedrine.

Full text of DOI:10.1016/0957-4166(96)00384-9

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