Synthesis of 2-aryltryptamines with palladium catalyzed cross-coupling of 2-bromotryptamines and arylboronic acids

DOI: 10.1016/S0040-4039(97)00797-1

Source and publish data:

Tetrahedron Letters p. 3871 - 3874 (1997)

Update date:2022-08-03

Topics:

Authors:

Chu, Lin

Fisher, Michael H.

Goulet, Mark T.

Wyvratt, Matthew J.

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1016/S0040-4039(97)00797-1

A versatile and high-yielding synthesis of 2-aryltryptamines employing palladium(0) catalyzed cross-coupling of 2-bromotryptamines and arylboronic acids was developed. The preparation of the intermediate 2-bromotryptamines with pyridine hydrobromide perbromide as the brominating agent, is also reported.

Full text of DOI:10.1016/S0040-4039(97)00797-1

Products guided by the article

Product name:1H-Isoindole-1,3(2H)-dione, 2-[2-[2-bromo-5-(phenylmethoxy)-1H-indol-3-yl]ethyl]-

Cas No:192182-48-2

R&D Labs maybe for 192182-48-2

ChangZhou Mascotchem. Co.,Ltd.

website:http://www.mascotchem.com

Contact:86-519-85010339

Address:B-802,XingBei Building,391#,Tongjiang Middle Road New District,Changzhou,JS,China
Nanjing Fubang Chemical Co.,Ltd

Contact:+86-25-83179199

Address:5F,Tianzheng international plaza,No399 Zhongyang Road ,Nanjing China
Kaymossy BioChem Tech Co., Ltd

website:http://www.kaimosi.com

Contact:0571-87191913/0571-87199097

Address:Room 215, Building 3rd, No.288 Ningxia Road, Qingdao city, China
Suzhou SuKaiLu Chemical Technology Co., Ltd.

Contact:+86-512-62766020

Address:Floor 4, Building 1, Xinyi Pharmaceutical Valley Wisdom Industrial Park, 415 Changyang Street, Suzhou Industrial Park, Jiangsu Province
Suzhou SuKaiLu Chemical Technology Co., Ltd.

Contact:+86-512-62766020

Address:Floor 4, Building 1, Xinyi Pharmaceutical Valley Wisdom Industrial Park, 415 Changyang Street, Suzhou Industrial Park, Jiangsu Province

Relevant to this article

Synthesis of (1R,4S,6R)-5,5,6-trimethyl-2-phosphabicyclo[2.2.2]octane and derivatives

Doi:10.1039/b924983d
(2010)
Asymmetric Construction of Cyclobutanes via Direct Vinylogous Michael Addition/Cyclization of β,γ-Unsaturated Amides

Doi:10.1021/acs.orglett.0c02488
(2020)
Cationic complexes of antimony(III) and bismuth(III) stabilized by intra- or intermolecular coordination

Doi:10.1021/om970322k
(1997)
Enantiospecific total synthesis of the potent antitumor macrolides cryptophycins 1 and 8

Doi:10.1021/jo971645t
(1997)
Synthesis and cytotoxicity of amino analogues of the potent DNA alkylating agent seco-CBI-TMI

Doi:10.1016/S0960-894X(97)00259-X
(1997)
Asymmetric Synthesis of (-)-Denticulatins A and B via Group-Selective Aldolization of a Meso Dialdehyde with a Chiral N-Propionylsultam.

Doi:10.1016/0040-4039(95)00787-D
(1995)

Article Doi