Synthesis of 2-aryltryptamines with palladium catalyzed cross-coupling of 2-bromotryptamines and arylboronic acids

DOI: 10.1016/S0040-4039(97)00797-1

Source and publish data:

Tetrahedron Letters p. 3871 - 3874 (1997)

Update date:2022-08-03

Topics:

Authors:

Chu, Lin

Fisher, Michael H.

Goulet, Mark T.

Wyvratt, Matthew J.

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Article abstract of DOI:10.1016/S0040-4039(97)00797-1

A versatile and high-yielding synthesis of 2-aryltryptamines employing palladium(0) catalyzed cross-coupling of 2-bromotryptamines and arylboronic acids was developed. The preparation of the intermediate 2-bromotryptamines with pyridine hydrobromide perbromide as the brominating agent, is also reported.

Full text of DOI:10.1016/S0040-4039(97)00797-1

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