Synthesis of 2-aryltryptamines with palladium catalyzed cross-coupling of 2-bromotryptamines and arylboronic acids

DOI: 10.1016/S0040-4039(97)00797-1

Source and publish data:

Tetrahedron Letters p. 3871 - 3874 (1997)

Update date:2022-08-03

Topics:

Authors:

Chu, Lin

Fisher, Michael H.

Goulet, Mark T.

Wyvratt, Matthew J.

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1016/S0040-4039(97)00797-1

A versatile and high-yielding synthesis of 2-aryltryptamines employing palladium(0) catalyzed cross-coupling of 2-bromotryptamines and arylboronic acids was developed. The preparation of the intermediate 2-bromotryptamines with pyridine hydrobromide perbromide as the brominating agent, is also reported.

Full text of DOI:10.1016/S0040-4039(97)00797-1

Products guided by the article

Product name:1H-Isoindole-1,3(2H)-dione, 2-[2-[2-bromo-5-(phenylmethoxy)-1H-indol-3-yl]ethyl]-

Cas No:192182-48-2

R&D Labs maybe for 192182-48-2

Kunshan Yalong Trading Co,.Ltd

Contact:86-512-57621185

Address:805-807 Room Hongqiao Mansion ,1088 West Qianjin Road, Kunshan, Jiangsu，China
Guangzhou Reachin Chemical Co., Ltd

Contact:+86-20-37087379 ext.604

Address:A122C-1, Tianyuan Plaza, 401 Tianyuan Rd., Tianhe, Guangzhou, China
Beijing Tianjia Chemical Science & Technology Co.,Ltd

Contact:86-0550-2392698

Address:No.388, Shiliang Road (East),
Shandong LuZhou Amino Acid Co., Ltd

Contact:86-539-2218025

Address:yishui economic and technical development zone zhenxing south road
JIANGXI AIFEIMU TECHNOLOGY CO.，LTD

Contact:+86-570-6040289

Address:FINECHEMICAL PARK,ZIBU TOWN,WANNIAN COUNTY,JIANGXI PROV.,CHINA,ZIP

Relevant to this article

Synthesis of (1R,4S,6R)-5,5,6-trimethyl-2-phosphabicyclo[2.2.2]octane and derivatives

Doi:10.1039/b924983d
(2010)
Asymmetric Construction of Cyclobutanes via Direct Vinylogous Michael Addition/Cyclization of β,γ-Unsaturated Amides

Doi:10.1021/acs.orglett.0c02488
(2020)
Cationic complexes of antimony(III) and bismuth(III) stabilized by intra- or intermolecular coordination

Doi:10.1021/om970322k
(1997)
Enantiospecific total synthesis of the potent antitumor macrolides cryptophycins 1 and 8

Doi:10.1021/jo971645t
(1997)
Synthesis and cytotoxicity of amino analogues of the potent DNA alkylating agent seco-CBI-TMI

Doi:10.1016/S0960-894X(97)00259-X
(1997)
Asymmetric Synthesis of (-)-Denticulatins A and B via Group-Selective Aldolization of a Meso Dialdehyde with a Chiral N-Propionylsultam.

Doi:10.1016/0040-4039(95)00787-D
(1995)

Article Doi