Conformationally constrained no synthase inhibitors: Rigid analogs of L- N-iminoethylornithine

DOI: 10.1016/S0960-894X(98)00532-0

Source and publish data:

Bioorganic and Medicinal Chemistry Letters p. 2961 - 2966 (1998)

Update date:2022-09-26

Topics:

Authors:

Eustache, Jacques

Grob, Alfred

Lam, Charles

Sellier, Odile

Schulz, Gerhard

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1016/S0960-894X(98)00532-0

The synthesis of eight rigid analogs of L-N-iminoethylomithine (L-NIO) is described. The compounds have been evaluated for their inhibition of inducible nitric oxide synthase. Preliminary structure-activity relationships are discussed.

Full text of DOI:10.1016/S0960-894X(98)00532-0

Products guided by the article

Product name:(S)-Benzyloxycarbonylamino-((1S,3R)-3-hydroxy-cyclopentyl)-acetic acid methyl ester

Cas No:219558-32-4

R&D Labs maybe for 219558-32-4

Shanghai Gsyn Chemical Co.,Ltd.

Contact:86-021-67158290

Address:86-021-67158291
Hangzhou Ledun Technology Co.,Ltd.

Contact:86-571-18767088918

Address:No.6 street,XiaSha,Hangzhou,China.
Wuxi Pharma-Trading Import & Export Co.,Ltd.

Contact:+86-510-82304590 82716390

Address:Room 523,Youzu Alliance Building,No.88 Renmin Zhonglu,Wuxi,Jiangsu,China
Acros Pharmatech Limited

website:http://www.acrospharmatech.com

Contact:+1-3234804688

Address:Flat/RM 1502,Easey Commercial building 253-261 Hennessy Road,Wanchai，HongKong
Shandong Xinke Petrochemical Co., Ltd.

Contact:+86-546-7277016

Address:Gudao Industrial Park, Hekou District, Dongying, Shandong Province, China

Relevant to this article

Acid-Stable Ester Linkers for the Solid-Phase Synthesis of Immobilized Peptides

Doi:10.1002/cplu.202000246
(2020)
Preparation of silanediyl-bridged Fe-Fe and Fe-W dinuclear complexes. X- ray structures of [Cp*Fe(Co)(μ-CO) {μ-Si(H)CHPH₂}(CO)(n)MCp] (Cp* = C₅Me₅, Cp = C₅H₅, M = Fe, n = 1; M = W, n = 2)

Doi:10.1246/bcsj.71.2865
(1998)
Synthesis of diacylglycerol analogs of phosphatidylinositol 3,4,5- trisphosphate

Doi:10.1016/S0040-4039(98)02151-0
(1998)
Synthesis of 3,5-disubstituted 10,11-dihydro-5H-dibenz[b,f]azepines

Doi:10.1007/BF02539228
(1998)
2-amino-3-substituted-6-[(E)-1-phenyl-2-(N- methylcarbamoyl)vinyl]imidazo-[1,2-a]pyridines as a novel class of inhibitors of human rhinovirus: Stereospecific synthesis and antiviral activity

Doi:10.1021/jm9810405
(1999)
Angular benzobisthietes

Doi:10.1016/S0040-4039(98)02265-5
(1998)

Article Doi