Bioorganic and Medicinal Chemistry Letters p. 2625 - 2628 (1999)
Update date:2022-09-26
Topics:
Minami, Nathaniel K.
Reiner, John E.
Semple, J. Edward
Application of the Sharpless AD protocol to a series of α-(E)-benzylidene-δ-lactam precursors followed by selective deoxygenation provided efficient synthetic routes to the chiral quaternary α-hydroxy-γ-lactam derivatives 4 and 5. These functionalized intermediates and the diol precursors 3 are regarded as novel types of D-Phe-Pro dipeptide surrogates that are useful as enzyme active site probes.
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