European Journal of Medicinal Chemistry p. 1005 - 1016 (2018)
Update date:2022-09-26
Topics: Scaffold Thiadiazine Inhibitor Selective Activity Proliferation DYRK1A Human Lead
Kumar, Kunal
Man-Un Ung, Peter
Wang, Peng
Wang, Hui
Li, Hailing
Andrews, Mary K.
Stewart, Andrew F.
Schlessinger, Avner
DeVita, Robert J.
The Dual-Specificity Tyrosine Phosphorylation-Regulated Kinase 1A (DYRK1A) is an enzyme that has been implicated as an important drug target in various therapeutic areas, including neurological disorders (Down syndrome, Alzheimer's disease), oncology, and
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