Facile synthesis of 9-(arenethenyl)purines via Heck reaction of 9-vinylpurines and aryl halides

DOI: 10.1016/j.tetlet.2007.08.008

Source and publish data:

Tetrahedron Letters p. 7388 - 7391 (2007)

Update date:2022-08-02

Topics:

Authors:

Huang, Wei-Sheng

Wang, Yihan

Sundaramoorthi, Raji

Thomas, R. Mathew

Wen, David

Liu, Shuangying

Lentini, Scott P.

Das, Sasmita

Banda, Geetha

Sawyer, Tomi K.

Shakespeare, William C.

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1016/j.tetlet.2007.08.008

The first example of a Heck reaction with 9-vinylpurines and aryl halides is described. It gives exclusively E-9-(arenethenyl)purines in high yields. Subsequent hydrogenation furnishes 9-(arenethyl)purines quantitatively.

Full text of DOI:10.1016/j.tetlet.2007.08.008

Products guided by the article

Product name:C₂₂H₂₃N₆OP

Cas No:956733-06-5

R&D Labs maybe for 956733-06-5

Guangzhou Swan Chemical Co., Ltd.

Contact:+86-20-31075659

Address:NO.301, Hong ba fang investment BLDG 1,Guan chong village,Shiqi town,Panyu district,Guangzhou
SHAANXI TOP PHARM CHEMICAL CO.LTD

Contact:+86-029-85733403

Address:No.108 ,west sector,south er huan,xi'an,china
Yancheng Creator Chemical Co., Ltd

Contact:0086-515-88710008 88710068 88710858 88710868

Address:No.21 Renming Road, Longgang Town, Yandu County,Yancheng City
FOSHAN NANHAI ZHONGNAN PHARMACEUTICAL FACTORY

Contact:0086-0757-85609331

Address:XIAHENGTIAN INDUSTRIAL ZONE,SHAYONG VILLAGE,LISHUI TOWN
Nanjing Yuance Industry&Trade Co., Ltd.

website:http://www.njyuance.cn/

Contact:+86-25-85439097

Address:B1702, Aoti Bldg, No. 130, Aoti Avenue, Nanjing, China

Relevant to this article

Chemoenzymatic synthesis of d-biotin intermediate lactone via lipase-catalyzed desymmetrization of meso diols

Doi:10.1016/j.molcatb.2013.09.014
(2013)
Effective synthesis of cyclic carbonates from carbon dioxide and epoxides by phosphonium iodides as catalysts in alcoholic solvents

Doi:10.1016/j.tetlet.2013.10.068
(2013)
One-Pot, Three-Component Assembly of Indoloquinolines: Total Synthesis of Isocryptolepine

Doi:10.1021/acs.joc.6b03084
(2017)
Synthesis of a tin(II) 1,3-benzobis(thiophosphinoyl)methanediide complex and its reactions with aluminum compounds

Doi:10.1021/om300345u
(2012)
Discovery of 6-phenylimidazo[2,1-b]thiazole derivatives as a new type of FLT3 inhibitors

Doi:10.1016/j.bmcl.2015.08.068
(2015)
Synthesis of substituted azulenes via Pt(II)-Catalyzed ring-expanding cycloisomerization

Doi:10.1021/ol502270q
(2014)

Article Doi