Novel regioselective N-alkylations of 5-substituted-2H-tetrazoles

DOI: 10.1016/S0040-4039(00)98819-1

Source and publish data:

Tetrahedron Letters p. 1925 - 1928 (1990)

Update date:2022-08-15

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Authors:

Prhavc Prhavc

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Article abstract of DOI:10.1016/S0040-4039(00)98819-1

Regioselective alkylation of 5-substituted-2H-tetrazoles 1 to 2-alkyl derivatives 3 was achieved via decarboxylative alkylation with alkyl cyanoformates. Lesser selectivity was observed with chloroformates.

Full text of DOI:10.1016/S0040-4039(00)98819-1

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