Synthesis and structure-activity relationships of dynorphin A-(1-8) amide analogues

DOI: 10.1021/jm00163a034

Source and publish data:

Journal of Medicinal Chemistry p. 206 - 212 (1990)

Update date:2022-09-26

Topics:

Authors:

Yoshino Yoshino

Nakazawa

Arakawa Arakawa

Kaneko Kaneko

Tsuchiya

Matsunaga

Araki Araki

Ikeda Ikeda

Yamatsu Yamatsu

Tachibana

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Article abstract of DOI:10.1021/jm00163a034

In order to study the structure-activity relationships of dynorphin A-(1-8) amide [Dyn(1-8)-NH₂], 20 analogues were synthesized by the solution method. Their biological activities were determined in the three bioassays [guinea pig ileum (GPI),

Full text of DOI:10.1021/jm00163a034

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