A CONVERGENT SYNTHESIS OF A NOVEL NON-PEPTIDYL GROWTH HORMONE SECRETAGOGUE, L-692,429

DOI: 10.1016/0040-4039(95)02033-0

Source and publish data:

Tetrahedron Letters p. 9445 - 9448 (1995)

Update date:2022-07-29

Topics:

Authors:

Bhupathy, M.

Bergan, J. J.

McNamara, J. M.

Volante, R. P.

Reider, P. J.

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Article abstract of DOI:10.1016/0040-4039(95)02033-0

A practical, convergent synthesis of L-692,429 (1) from three key intermediates - the 3-aminobenzlactam 2, the β-lactam 3 and the biphenyltetrazole 4 - is described.The mechanism of the coupling reaction in which 3 is used as a β-aminoacid equivalent is a

Full text of DOI:10.1016/0040-4039(95)02033-0

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