A CONVERGENT SYNTHESIS OF A NOVEL NON-PEPTIDYL GROWTH HORMONE SECRETAGOGUE, L-692,429

DOI: 10.1016/0040-4039(95)02033-0

Source and publish data:

Tetrahedron Letters p. 9445 - 9448 (1995)

Update date:2022-07-29

Topics:

Authors:

Bhupathy, M.

Bergan, J. J.

McNamara, J. M.

Volante, R. P.

Reider, P. J.

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1016/0040-4039(95)02033-0

A practical, convergent synthesis of L-692,429 (1) from three key intermediates - the 3-aminobenzlactam 2, the β-lactam 3 and the biphenyltetrazole 4 - is described.The mechanism of the coupling reaction in which 3 is used as a β-aminoacid equivalent is a

Full text of DOI:10.1016/0040-4039(95)02033-0

Products guided by the article

Product name:(1,1-Dimethyl-2-{(R)-2-oxo-1-[2'-(2-trityl-2H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-2,3,4,5-tetrahydro-1H-benzo[b]azepin-3-ylcarbamoyl}-ethyl)-sulfamic acid methyl ester

Cas No:174222-36-7

R&D Labs maybe for 174222-36-7

QINGDAO NEW FLOURISH INTERNATIOANAL TRADE CO., LTD.

Contact:+86 532 80861829

Address:No. 1, Yinchuan East Road, 266061, Qingdao, China
Jiangsu Fengshan Group Co., Ltd.

Contact:86-25-86558671

Address:1903,Central International Mansion 105-6 North Zhongshan Road, Nanjing, China
Leshan Kai Yada Photoelectric Technology Co., Ltd.,

website:http://www.kydmaterials.com

Contact:0833-5603116

Address:Airport road Jiajiang county, Sichuan province,China
Taimai Sanluck Pharmaceutical Co.,Ltd

Contact:86-592-7662921

Address:8D,No.186,Huarong Road,Huli,Xiamen,China
Shanghai Yuanding Chem. Sci. & Tech. Co., Ltd.

website:http://www.shydtec.com

Contact:86-21-57721279

Address:Science and Technology Park, Songjiang District, Shanghai, China

Relevant to this article

Doi:10.1021/jm00307a016
(1968)
An Intramolecular Diels-Alder Approach to Tricyclic Taxoid Skeletons

Doi:10.1016/S0040-4039(00)79157-X
(1993)
Studies towards the synthesis of (+)-ptilomycalin A; stereoselective N-acyliminium ion coupling reactions to enantiopure C-2 substituted lactams

Doi:10.1016/0040-4020(95)01085-8
(1996)
The preparation of substituted 3,4-dihydro-1(2H)-naphthalenones from benzocyclobutenones via sequential thermal electrocyclic reactions

Doi:10.1016/0040-4020(95)01054-8
(1996)
Synthesis of Microcolin B, a Potent New Immunosuppressant Using an Efficient Mixed Imide Formation Reaction

Doi:10.1021/jo970387x
(1997)
A New Powerful and Practical BLA Catalyst for Highly Enantioselective Diels-Alder Reaction: An Extreme Acceleration of Reacrion Rate by Broensted Acid

Doi:10.1021/ja954060u
(1996)

Article Doi