Amino acids and peptides. LIII. Synthesis and biological activities of some pseudo-peptide analogs of PKSI-527, a plasma kallikrein selective inhibitor: The importance of the peptide backbone

DOI: 10.1248/cpb.47.1141

Source and publish data:

Chemical and Pharmaceutical Bulletin p. 1141 - 1144 (1999)

Update date:2022-08-02

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Authors:

Fukumizu, Atsuko

Tsuda, Yuko

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Article abstract of DOI:10.1248/cpb.47.1141

Pseudo-peptide analogs of trans-4-aminomethylcyclohexanecarbonyl-L- phenylalanyl-4-aminophenyl acetic acid (PKSI-527, plasma kallikrein selective inhibitor), in which an amide bond (peptide bond) has been replaced by a CH₂-NH bond, i.e. trans-4

Full text of DOI:10.1248/cpb.47.1141

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