Amino acids and peptides. LIII. Synthesis and biological activities of some pseudo-peptide analogs of PKSI-527, a plasma kallikrein selective inhibitor: The importance of the peptide backbone

DOI: 10.1248/cpb.47.1141

Source and publish data:

Chemical and Pharmaceutical Bulletin p. 1141 - 1144 (1999)

Update date:2022-08-02

Topics:

Authors:

Fukumizu, Atsuko

Tsuda, Yuko

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1248/cpb.47.1141

Pseudo-peptide analogs of trans-4-aminomethylcyclohexanecarbonyl-L- phenylalanyl-4-aminophenyl acetic acid (PKSI-527, plasma kallikrein selective inhibitor), in which an amide bond (peptide bond) has been replaced by a CH₂-NH bond, i.e. trans-4

Full text of DOI:10.1248/cpb.47.1141

NII-Electronic Library Service

Products guided by the article

Product name:Boc-Tra-L-Phe-ψ(CH2-NH)-APAA-OBzl

Cas No:248953-94-8

R&D Labs maybe for 248953-94-8

Shanghai Bojing Chemical Co., Ltd.

Contact:021-37122233

Address:6F Buildiing 11,No.388,Baifu Road,District Fengxian.Shanghai, China.
Rayfull Holding Co., Ltd

Contact:+86-577-65618087-605

Address:Room 402, Unit 4 Xinhu Bldg. Waitan Ruian City, Zhejiang China.
HEZE KINGVOLT CHEMICAL CO., LTD

Contact:86-573-82118911

Address:Juancheng Industry Park
Synasia Inc

Contact:17316303296

Address:240 Amboy Ave
Wuhan Yitongtai Science and Technology Co.,Ltd.

Contact:+86-27-88933550

Address:27th Fl. Bldg. 1, Shuian International Mansion, Heping Ave, Wuhan, Hubei, China

Relevant to this article

Synthesis, characterization, and reactivity of titanium(IV) complexes supported by proximally bridged p-tert-butylcalix[4]arene ligands

Doi:10.1016/S0022-328X(99)00279-X
(1999)
The Triazene Moiety as a Protecting Group for Aromatic Amines

Doi:10.1021/jo00060a028
(1993)
Recycling of homogeneous catalysts in reactive ionic liquid-solvent-free aminofunctionalizations of alkenes

Doi:10.1039/c7gc02272g
(2017)
Selective solid-phase iodination of phenolic groups with bis(pyridine)iodonium (I) tetrafluoroborate

Doi:10.1016/S0040-4039(99)01522-1
(1999)
Reaction of polyhalo semiquinoid structures originating from 4-aroyl(arylsulfonyl)oximino-2,5-cyclohexadiene-1-ones with arylsulfinic acids

Doi:10.1023/A:1012395400078
(2001)
2,2,4,4,6,6-Hexabenzylcyclotristannatellurane, (Bn₂SnTe)₃. Synthesis and Structural Characterization of an Organometallic Single-Source Precursor to Phase-Pure, Polycrystalline SnTe

Doi:10.1021/om990506u
(1999)

Article Doi