Preparation of N-phosphorylated nitrogen mustards with the benzodiaza-and oxazaphosphorinone ring systems; hydrolysis of 2-chloro benzodiazaphosphorinones

Article abstract of DOI:10.1080/10426509608046400

The reaction of N-p-ethoxyphenylanthranilic acid 1 with phosphorus trichloride furnished the 2-chloro-1,3,2-benzoxazaphosphorin-6-one 2, which was allowed to react with bis-(2-chloroethyl)amine hydrochloride to form 3 by substitution at phosphorus. Treatm

Full text of DOI:10.1080/10426509608046400

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Phosphorus, Sulfur, and Silicon and the
Related Elements
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PREPARATION OF N-PHOSPHORYLATED
NITROGEN MUSTARDS WITH
THE BENZODIAZA- AND
OXAZAPHOSPHORINONE RING
SYSTEMS;HYDROLYSIS OF 2-CHLORO
BENZODIAZAPHOSPHORINONES
Ion Neda a , Ralf Sonnenburg a , Axel Fischer a , Peter G. Jones a
Reinhard Schmutzler a
&
a Institut für Anorganische und Analytische Chemie der Technischen
Universität , Postfach 3329, D-38023, Braunschweig, Germany
Published online: 04 Oct 2006.
To cite this article: Ion Neda , Ralf Sonnenburg , Axel Fischer , Peter G. Jones & Reinhard
Schmutzler (1996) PREPARATION OF N-PHOSPHORYLATED NITROGEN MUSTARDS WITH
THE BENZODIAZA- AND OXAZAPHOSPHORINONE RING SYSTEMS;HYDROLYSIS OF 2-CHLORO
BENZODIAZAPHOSPHORINONES, Phosphorus, Sulfur, and Silicon and the Related Elements, 113:1-4,
287-294, DOI: 10.1080/10426509608046400
To link to this article: http://dx.doi.org/10.1080/10426509608046400
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